Concise Synthesis of Densely Substituted
Azaheterocycles
Dr. Mohammad Movassaghi, Assistant Professor, Massachusetts Institute of Technology, Department of Chemistry, Cambridge, MA, USA
A series of new methodologies will be discussed that enable the concise synthesis of a variety of azaheterocycles from readily available starting materials. A key aspect of these methodologies is the electrophilic activation of amides for nucleophilic trapping by a variety of sigma and pi-nucleophiles.